Clinical / Pharmaceutical

Tetracosactide

Cosyntropin · Synacthen · ACTH 1-24 · Tetracosactrin

Tetracosactide (Cosyntropin) is the pure, synthetic recreation of the first 24 amino acids of the human Adrenocorticotropic Hormone (ACTH) - the exact sequence holding 100% of the molecule's biological firepower. It is the absolute clinical standard for aggressive diagnostic interrogation of the adrenal glands, utilized instantly in emergency and endocrine settings to forcefully test the maximum acute cortisol-producing capacity of a failing adrenal cortex.

Not FDA-approved - research chemical
Reviewed by CalcMyPeptide Editorial Team
Last updated: August 2026Evidence: High1 peer-reviewed citation
Typical research dose
250 mcg IV/IM (diagnostic)
Frequency
Single dose (ACTH stimulation test)
Half-life
~15-20 minutes
Common vials
N/A (oral)
CAS
16960-16-0
Molecular weight
2933.5 g/mol

Use-case scores

0–10 against the evidence we have, not a gym ranking. Hidden domains do not apply here.

  • Sexual / hormonal3/10

    Diagnostic ACTH analog. Not a tan peptide and not a gym cortisol hack.

Compound card

Class
ACTH(1-24) (cosyntropin / Synacthen diagnostic)
Formula
C136H210N40O31S
Status
Not FDA-approved · research use

How it works

Tetracosactide (also known as cosyntropin or Synacthen) is a synthetic peptide consisting of the first 24 amino acids of adrenocorticotropic hormone (ACTH). The full human ACTH has 39 amino acids, but biological activity resides entirely in the N-terminal 24 sequence.

Tetracosactide stimulates the adrenal cortex to rapidly produce cortisol and other corticosteroids. It is primarily used clinically as a rapid diagnostic test (the Synacthen Test) for adrenal insufficiency. Unlike long-term corticosteroid therapy, it relies on the body's own adrenal steroidogenic pathways.

Source: PMID: 6765449

Background & History

Tetracosactide (cosyntropin/Synacthen) is an essential diagnostic tool in endocrinology. The ACTH stimulation test has been the gold standard for diagnosing adrenal insufficiency for over 50 years. The short Synacthen test takes only 1 hour and can be performed in outpatient settings. Depot formulations (Synacthen Depot) have also been used therapeutically for infantile spasms and inflammatory conditions in various countries.

Research Use Cases

  • ✓Adrenal insufficiency diagnosis
  • ✓ACTH stimulation test
  • ✓Infantile spasms (depot form)
  • ✓Therapeutic use in inflammatory conditions

Dosing

PhaseDoseFrequencyNotes
Diagnostic (Synacthen Test)250 mcgSingle IV or IM doseFDA-approved diagnostic standard for adrenal insufficiency.
Therapeutic (Rare)1 mg DepotVariesUsed rarely in cases like infantile spasms or MS exacerbations where endogenous cortisoid release is preferred over oral steroids.

Administration

Route / form
IV or IM injection
Timing
Morning (diagnostic test).
Empty stomach?
No - Food timing is not critical.

Timeline

30-60 minutes
Diagnostic blood draw for peak cortisol response. Cortisol should rise above 18-20 μg/dL.

Who it is for

Adrenal Function Testing

High

The gold-standard diagnostic tool for Addison's disease and HPA axis evaluation.

Safety & Considerations

FDA-approved. Mostly used in supervised clinical settings for single-dose diagnosis. Therapeutic use carries risks similar to chronic corticosteroid exposure.

Regulatory & Legal Status

FDA Status (US)
Research Only
WADA Status (2026)
Not Listed

Not currently on the WADA 2026 Prohibited List. Policies may change - verify before competition.

Classification

Research Chemical

US Compounding: Not eligible / not available

⚠️ This information is for educational purposes only and may not reflect the most current regulatory updates. Always verify with official FDA, WADA, and jurisdiction-specific sources before use.

Limits of current evidence

  • Not a pigmentation protocol.

Verdict

Tetracosactide is cosyntropin. The 250 mcg stim test is endocrinology. It is not MT-2. Stimulating cortisol on purpose without a clinic is a bad idea.

Interactions & Contraindications

Exogenous corticosteroids will blunt the cortisol response and should be withheld before testing. Dexamethasone does not cross-react with cortisol assays.

Frequently Asked Questions

What is the Synacthen test?▼
It is a diagnostic test where tetracosactide (synthetic ACTH) is injected, and your cortisol is measured 30-60 minutes later. If cortisol does not rise adequately, it indicates primary adrenal insufficiency (Addison's disease).

References

  1. Dorin RI et al. “"The standard short Synacthen test in adrenal insufficiency".” Annals of Internal Medicine (2003). PMID: 12860585

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