CalcMyPeptide
Healing & RecoveryAlso known as: Vasoactive Intestinal Peptide

VIP

Vasoactive Intestinal Peptide (VIP) is an endogenous 28-amino-acid neuropeptide that reigns as the master regulator of systemic immunity and vascular tone. In elite functional medicine, VIP is the definitive, heavy-artillery intervention for crippling autoimmune cascades, specifically Chronic Inflammatory Response Syndrome (CIRS) triggered by toxic mold (mycotoxins) or catastrophic severe post-viral syndromes. Deployed primarily via nasal spray, it rapidly arrests systemic cytokine storms, restores severely compromised pulmonary function, and violently reverses neuroinflammation.

Reviewed by CalcMyPeptide Editorial Team
Last updated: April 2026Evidence: Moderate2 peer-reviewed citations

Quick Stats

Half-Life~2 minutes (IV); longer with intranasal
Dose Range50-200 mcg (intranasal)
Frequency1-2× daily (intranasal)
Vial SizesN/A (oral)
BioavailabilityIntranasal spray (preferred) or IV
Year Developed1970

Scientific Data

Molecular Formula
C147H237N43O43S1
Molecular Weight
3326.79 g/mol
CAS Number
PubChem ID
Developer
Said SI, Mutt V (isolated from porcine intestine)

Mechanism of Action

VIP (Vasoactive Intestinal Peptide) is a 28-amino-acid regulatory neuropeptide that acts through VPAC1 and VPAC2 receptors. It exerts potent vasodilatory, anti-inflammatory, bronchodilatory, and immunomodulatory effects throughout the body.

VIP plays a critical role in pulmonary homeostasis — regulating airway smooth muscle tone, pulmonary arterial pressure, and local immune responses. It has been studied extensively for Chronic Inflammatory Response Syndrome (CIRS/mold illness), post-COVID immune dysregulation, and mast cell activation syndrome (MCAS). In the Shoemaker CIRS protocol, VIP is administered intranasally as the final restoration step — addressing residual pulmonary inflammation and normalizing inflammatory markers (VEGF, TGF-β1, MMP-9) after upstream biotoxin treatment. VIP also has neuroprotective and circadian-regulatory properties.

Source: PMID: 15271596

Background & History

VIP (Vasoactive Intestinal Peptide) is a 28-amino-acid neuropeptide discovered in 1970 by Said and Mutt in porcine intestinal tissue. It functions as both a neurotransmitter and hormone, with receptors VPAC1 and VPAC2 distributed throughout the CNS, GI tract, lungs, and immune system. VIP is one of the most potent endogenous anti-inflammatory neuropeptides known, with emerging roles in autoimmune disease, pulmonary arterial hypertension, and chronic inflammatory conditions including MCAS and Long COVID.

Research Use Cases

  • Chronic inflammatory conditions: MCAS, CIRS, Long COVID
  • Pulmonary arterial hypertension (PAH)
  • Autoimmune regulation: rheumatoid arthritis, Crohn's, MS research
  • Gastrointestinal motility disorders
  • Neuroprotection in Parkinson's and Alzheimer's (preclinical)

Dosing Protocol

Typical Dose50-200 mcg (intranasal)
Frequency1-2× daily (intranasal)
Half-Life~2 minutes

Dosing Protocols

Shoemaker CIRS Protocol

Dose
50 mcg
Frequency
4x daily intranasal (each nostril)
Note: Standard Shoemaker CIRS protocol. Must complete upstream treatment steps before VIP. Monitor VEGF and TGF-β1 labs throughout.

General Immunomodulation

Dose
50 - 200 mcg
Frequency
1-3x daily intranasal
Note: For pulmonary inflammation, post-COVID dysregulation, and MCAS. Lower doses for general use.

Body-Weight Dosing Reference

Estimated doses extrapolated from the published research range of 50200 mcg/day (referenced to 70 kg / 154 lb). These are approximations — consult a qualified healthcare provider for personalised guidance.

WeightLowTargetHigh
120 lb(54 kg)39 mcg96 mcg154 mcg
140 lb(63 kg)45 mcg113 mcg180 mcg
160 lb(73 kg)52 mcg130 mcg209 mcg
180 lb(82 kg)59 mcg146 mcg234 mcg
200 lb(91 kg)65 mcg163 mcg260 mcg
220 lb(100 kg)71 mcg179 mcg286 mcg
250 lb(113 kg)81 mcg202 mcg323 mcg

💉 For exact syringe units based on your vial concentration, use the VIP Reconstitution Calculator →

Administration

Route
Intranasal spray
Timing
Spread doses throughout the day. No fasting required.
Fasting Required?
No — food timing not critical

Expected Timeline

Week 1-2
Improved breathing and reduced pulmonary symptoms. Inflammatory markers begin normalizing.
Week 4-8
VEGF, TGF-β1, MMP-9 normalization in CIRS protocol. Improved cognitive and physical function.

Who Is It For?

CIRS / Mold Illness

Moderate

Final step in Shoemaker protocol. Addresses residual pulmonary inflammation after biotoxin pathway treatment.

Post-COVID Immune Dysregulation

Low

Studied for long-COVID inflammatory patterns. Emerging evidence for immunomodulatory benefit.

Pulmonary Hypertension

Low

Research suggests VIP deficiency in pulmonary arterial hypertension. IV VIP trials show promise.

Safety & Considerations

Research peptide used clinically in CIRS protocols. Primarily administered intranasally. May cause transient vasodilation (facial flushing, mild hypotension). Not for use in patients with active diarrhea. Monitor blood pressure with initial doses.

Regulatory & Legal Status

FDA Status (US)
Research Only
WADA Status (2026)
Not Listed

Not currently on the WADA 2026 Prohibited List. Policies may change — verify before competition.

Classification

Research Chemical

US Compounding: Not eligible / not available

⚠️ This information is for educational purposes only and may not reflect the most current regulatory updates. Always verify with official FDA, WADA, and jurisdiction-specific sources before use.

Interactions & Contraindications

Potent vasodilator — risk of blood pressure drop, especially with concurrent antihypertensive medications. Very short half-life (1-2 min) requires intranasal or continuous IV administration. Compounded intranasal VIP is most common route in CIRS protocols.

Synergies & Common Stacks

VIP provides broad anti-inflammatory signaling; BPC-157 handles specific tissue repair post-inflammation. Comprehensive for inflammatory GI conditions.

VIP modulates the immune system centrally; KPV blocks NF-κB locally. Together address inflammation from systemic and cellular levels.

Dosing Quick Reference

VIP— Dosing Guide
Dose Range
50-200 mcg (intranasal)
Half-Life
~2 minutes
Frequency
1-2× daily (intranasal)
Route
Intranasal
Healing & Recoverycalcmypeptide.com

Frequently Asked Questions

What is VIP used for in CIRS?
VIP is the final step in the Shoemaker CIRS protocol, addressing pulmonary inflammation, reducing inflammatory markers (VEGF, TGF-β1, MMP-9), and restoring normal immune regulation. It must be administered intranasally AFTER upstream biotoxin pathway steps are completed.
How is VIP administered?
Primarily intranasal — 50 mcg per nostril, 4x daily in the Shoemaker protocol. Intranasal delivery provides direct CNS/pulmonary access. IV is reserved for research settings.

References

  1. Shoemaker RC et al. "Restoration of inflammatory markers in CIRS with intranasal VIP".” Internal Medicine Review (2017). PMID: 28694751
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