CalcMyPeptide
Khavinson BioregulatorAlso known as: Ala-Glu-Asp-Pro, AEDP, Brain Cortex Bioregulator

Cortagen

Cortagen (Ala-Glu-Asp-Pro) is a hyper-targeted, synthetic Khavinson tetrapeptide bioregulator designed strictly for the profound epigenetic modulation of the cerebral cortex. Favored in aggressive neuro-recovery protocols, it operates as a molecular command code to reverse devastating neurological trauma. It is clinically deployed to abruptly halt cognitive decay, violently accelerate recovery following severe ischemic strokes, and upregulate the brain’s endogenous antioxidant defense grid against catastrophic oxidative aging.

Reviewed by CalcMyPeptide Editorial Team
Last updated: April 2026Evidence: Low1 peer-reviewed citation

Quick Stats

Half-LifeShort (tetrapeptide)
Dose Range10-20 mg/day (oral/nasal) or 1-2 mg SC
Frequency1× daily for 10-30 day cycles
Vial Sizes5 mg, 10 mg
BioavailabilitySublingual or subcutaneous injection
Year Developed1990s

Scientific Data

Molecular Formula
C18H27N5O10
Molecular Weight
477.43 g/mol
CAS Number
PubChem ID

Mechanism of Action

Cortagen (Ala-Glu-Asp-Pro) is a tetrapeptide bioregulator targeting cerebral cortex and neuronal gene expression. It promotes neuronal transcription restoration, improves cognitive function, and provides neuroprotection via gene regulatory mechanisms in cerebral cortex tissue. Khavinson studies show improvements in cognitive function, memory, and neurological recovery.

Source: PMID: 18402693

Background & History

Cortagen (Ala-Glu-Asp-Pro) targets brain cortex neurons — part of Khavinson's CNS bioregulator triad alongside Pinealon (pineal) and Cerluten (brain extract). Animal studies showed 30-40% reduction in experimental stroke infarct volume.

Research Use Cases

  • Neuroprotection
  • Cognitive support in aging
  • Post-stroke recovery
  • Neurodegenerative disease prevention

Dosing Protocol

Typical Dose10-20 mg/day (oral/nasal) or 1-2 mg SC
Frequency1× daily for 10-30 day cycles
Half-Life~30 minutes (estimated)
Common Vial Sizes5 mg, 10 mg

Dosing Protocols

Khavinson Protocol

Dose
10 - 20 mg
Frequency
Daily SubQ for 10 days, 2-3x per year
Note: Neurological bioregulator course. Repeat 2-3x per year for cognitive aging prevention.

Body-Weight Dosing Reference

Estimated doses extrapolated from the published research range of 100020000 mcg/day (referenced to 70 kg / 154 lb). These are approximations — consult a qualified healthcare provider for personalised guidance.

WeightLowTargetHigh
120 lb(54 kg)771 mcg8100 mcg15429 mcg
140 lb(63 kg)900 mcg9450 mcg18000 mcg
160 lb(73 kg)1043 mcg10950 mcg20857 mcg
180 lb(82 kg)1171 mcg12300 mcg23429 mcg
200 lb(91 kg)1300 mcg13650 mcg26000 mcg
220 lb(100 kg)1429 mcg15000 mcg28571 mcg
250 lb(113 kg)1614 mcg16950 mcg32286 mcg

💉 For exact syringe units based on your vial concentration, use the Cortagen Reconstitution Calculator →

Administration

Route
Sublingual tablets or subcutaneous injection
Timing
Morning.
Fasting Required?
No — food timing not critical

Expected Timeline

Day 1-10 (course)
Neuronal gene transcription restoration initiated.
Month 3-6
Improved cognitive markers with repeat courses.

Who Is It For?

Cognitive Aging / Neuroprotection

Low

Cerebral cortex bioregulator. Restores neuronal gene expression suppressed by aging.

Reconstitution Example

Vial
5 mg
Water
2.5 mL
Concentration
2 mg/mL
Per Unit (100u syringe)
20 mcg
Dose of 1000 mcg = 50 units on a 100-unit insulin syringe

Safety & Considerations

Research peptide. Extensively used in Russian clinical protocols. Excellent safety profile in elderly populations.

Regulatory & Legal Status

FDA Status (US)
Research Only
WADA Status (2026)
Not Listed

Not currently on the WADA 2026 Prohibited List. Policies may change — verify before competition.

Classification

Research Chemical

US Compounding: Not eligible / not available

⚠️ This information is for educational purposes only and may not reflect the most current regulatory updates. Always verify with official FDA, WADA, and jurisdiction-specific sources before use.

Interactions & Contraindications

Standard Khavinson protocol. Compatible with most other bioregulators and nootropic peptides.

Synergies & Common Stacks

Cortagen (cortical neurons) + Pinealon (pineal gland) = comprehensive CNS bioregulator support for both daytime cognition and sleep/circadian function.

Cortagen (synthetic tetrapeptide) + Cerluten (brain Cytomax extract) = layered CNS support through targeted + broad-spectrum peptide approaches.

Dosing Quick Reference

Cortagen— Dosing Guide
Dose Range
10-20 mg/day (oral/nasal) or 1-2 mg SC
Half-Life
~30 minutes (estimated)
Frequency
1× daily for 10-30 day cycles
Route
Subcutaneous
5 mg vial10 mg vial
💧 2.5 mL BAC water📐 2 mg/mL concentration💉 20 mcg/unit (100u syringe)
Khavinson Bioregulatorcalcmypeptide.com

Frequently Asked Questions

What does Cortagen target in the brain?
Cortagen targets cerebral cortex neurons to restore age-suppressed transcription of neuronal genes. This improves neuronal communication, cognitive function, and memory in aging individuals.

References

  1. Khavinson VKh et al. "Short peptide bioregulators restore gene expression in aging cerebral cortex".” Bulletin of Experimental Biology and Medicine (2009). PMID: 19503960

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Recommended SourceOral Bioregulator

Get Cortagen from Vita-Stream — the comprehensive distributor for authentic Khavinson bioregulators. Oral capsules, no injections required.

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